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2017 Vol. 25, No. 2
Published: 20 February 2017

 
93 Design, Synthesis and Antitumor Activities of Novel Pyridine c-Met Kinase Inhibitors
SONG Ping, LI Jun-ming, QIN Ting-ting, CHANG Xian-lei, YANG Yang, LIANG Huan, ZHU Yu, ZHAO Yan-Jin, LI Shu-xin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16285
2017 Vol. 25 (2): 93-98 [Abstract] ( 324 ) HTML (1 KB)  PDF (2567 KB)  ( 250 )
99 Design, Synthesis and Biological Activities of Novel PARP-1 Inhibitors with Pyrazolotriazinone Skeleton
LIU Zhi-xiong, WANG Xiao-long, XUE Xin, LI Fu-wei, YU Hai-tao
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16280
2017 Vol. 25 (2): 99-106 [Abstract] ( 316 ) HTML (1 KB)  PDF (2943 KB)  ( 292 )
107 Synthesis of Novel Five-membered Carbocyclic Spirooxindoles and Their Activities Against Human Leukemia Cells
CHEN Zhi-yong, TIAN Min-yi, YANG Jun, LIU Huan-huan, LIN Bing, PAN Yu-jie, LIU Xiong-li
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16260
2017 Vol. 25 (2): 107-111 [Abstract] ( 331 ) HTML (1 KB)  PDF (1266 KB)  ( 313 )
112 N,N-Dimethylacetamide-promoted Synthesis of Cinnamyl Carboxylate and The Co-promoted Mechanism
ZHU Xian-hong, ZHOU An-xi, LUO Nian-hua, PENG Liang, ZENG Xian-zhu, ZHENG Da-gui
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16229
2017 Vol. 25 (2): 112-120 [Abstract] ( 303 ) HTML (1 KB)  PDF (2358 KB)  ( 626 )
121 “One-Pot” Synthesis of α,β-Alkynones Promoted by Magnesium Powder
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16264
2017 Vol. 25 (2): 121-126 [Abstract] ( 282 ) HTML (1 KB)  PDF (663 KB)  ( 312 )
127 Synthesis of p-Methoxyacetophenone Catalyzed by Molecular Sieve PW-β/MCM-41 Modified with Phosphotungstic Acid
JIAO Lei, LIU Han, LI Hui-peng, ZHAO Hua
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16177
2017 Vol. 25 (2): 127-131 [Abstract] ( 338 ) HTML (1 KB)  PDF (1485 KB)  ( 212 )
132 Hydrothermal Preparation of Chiolite-type Fluoride K5V3F14 and Its Magnetic Property
HE Li-jie, ZHANG Dong, TAN Guang-lei, MU Tao, LIU Hai-yan, DU Peng
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16129
2017 Vol. 25 (2): 132-136 [Abstract] ( 234 ) HTML (1 KB)  PDF (1225 KB)  ( 251 )
137 Solid-phase Synthesis of Polypeptides BRC4 and Their Interaction with RAD51(231-260)
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16216
2017 Vol. 25 (2): 137-139 [Abstract] ( 259 ) HTML (1 KB)  PDF (470 KB)  ( 239 )
140 Preparation of A Novel Degradable Anti-inflammatory Sustain Release System By Combination of Hot Melt Extrusion and Electrospining Method
WANG Lian-song, YIN Li-li, LIU Dong, ZHENG Yu-qiang, HE Wei
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16175
2017 Vol. 25 (2): 140-143 [Abstract] ( 280 ) HTML (1 KB)  PDF (811 KB)  ( 258 )
144 Synthesis of Methyl Laurate Catalyzed by Concerted Catalysis of TsOH Cooperate with I2
WANG Lin-lin, DU Ying, WU Xiao-yun, LUO Shi-xia, YIN Xiao-gang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16145
2017 Vol. 25 (2): 144-147 [Abstract] ( 249 ) HTML (1 KB)  PDF (686 KB)  ( 204 )
148 Synthesis of An End-hydroxy PAMAM Molecular
SHI Jun, GUO Xiao-yi, WANG Ru-bin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16242
2017 Vol. 25 (2): 148-151 [Abstract] ( 276 ) HTML (1 KB)  PDF (1004 KB)  ( 250 )
152 Analysis of Related Substances in The Production of Ursodeoxycholic Acid
XIE Qiang, WANG Kun, TAO Jia-lin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16279
2017 Vol. 25 (2): 152-154 [Abstract] ( 425 ) HTML (1 KB)  PDF (578 KB)  ( 295 )
155 Research on Selective Demethylation of Trimethoxybenzene Compounds
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16185
2017 Vol. 25 (2): 155-158 [Abstract] ( 262 ) HTML (1 KB)  PDF (846 KB)  ( 274 )
159 Microwave Synthesis of 4,7,10-Tris(tert-butoxycarbonylmethyl)-1,4,7,10-tetraazacyclodo-decane-1-acetohydrazide
ZHOU Jin, YANG Hai-dong, SUN Hong-shun, LI Yu-long, JIANG Hong
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16234
2017 Vol. 25 (2): 159-162 [Abstract] ( 257 ) HTML (1 KB)  PDF (1734 KB)  ( 312 )
163 Synthesis and Properties of Acrylamide/Methyl Acryloyl Oxygen Ethyl Dimethyl Ammonium Propyl Sulfonic Acid Copolymer
GUAN Hui-min, ZHAGN Wei-wei, YU Ting-yun
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16223
2017 Vol. 25 (2): 163-165 [Abstract] ( 260 ) HTML (1 KB)  PDF (788 KB)  ( 280 )
166 Process Improvement on the Synthesis of Afatinib
LI Wen-qian, SONG Guo-qiang, WAN Yi-dong, GAO You-jun, FENG Xiao-qing
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16253
2017 Vol. 25 (2): 166-169 [Abstract] ( 409 ) HTML (1 KB)  PDF (1343 KB)  ( 373 )
170 Process Improvement on Synthesis of Vitamin D2-A and CD Ring Fragment Alcohol
CHEN Guang-yao, BAO Xiao-zhen, DING Ying, ZHANG Heng-rui, FANG Zhi-jie
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16225
2017 Vol. 25 (2): 170-172 [Abstract] ( 274 ) HTML (1 KB)  PDF (573 KB)  ( 244 )
173 Research Progress on Synthesis of Acridine Derivatives
WEI Qiang, GENG Xin-le
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16288
2017 Vol. 25 (2): 173-177 [Abstract] ( 374 ) HTML (1 KB)  PDF (3739 KB)  ( 708 )
178 Research Progress on the Synthesis and Bioactivities of Indole-3-glyoxylamide Derivatives
HU Hong-yu, WANG Fei, ZHAO Sheng-xian, FANG Mei-juan
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16207
2017 Vol. 25 (2): 178-184 [Abstract] ( 362 ) HTML (1 KB)  PDF (2621 KB)  ( 263 )
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