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2017 Vol. 25, No. 2
Published: 20 February 2017
93
Design, Synthesis and Antitumor Activities of Novel Pyridine
c
-Met Kinase Inhibitors
SONG Ping, LI Jun-ming, QIN Ting-ting, CHANG Xian-lei, YANG Yang, LIANG Huan, ZHU Yu, ZHAO Yan-Jin, LI Shu-xin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16285
2017 Vol. 25 (2): 93-98 [
Abstract
] (
324
)
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(1 KB)
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(2567 KB) (
250
)
99
Design, Synthesis and Biological Activities of Novel PARP-1 Inhibitors with Pyrazolotriazinone Skeleton
LIU Zhi-xiong, WANG Xiao-long, XUE Xin, LI Fu-wei, YU Hai-tao
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16280
2017 Vol. 25 (2): 99-106 [
Abstract
] (
316
)
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(1 KB)
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(2943 KB) (
292
)
107
Synthesis of Novel Five-membered Carbocyclic Spirooxindoles and Their Activities Against Human Leukemia Cells
CHEN Zhi-yong, TIAN Min-yi, YANG Jun, LIU Huan-huan, LIN Bing, PAN Yu-jie, LIU Xiong-li
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16260
2017 Vol. 25 (2): 107-111 [
Abstract
] (
331
)
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(1 KB)
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(1266 KB) (
313
)
112
N,N-
Dimethylacetamide-promoted Synthesis of Cinnamyl Carboxylate and The Co-promoted Mechanism
ZHU Xian-hong, ZHOU An-xi, LUO Nian-hua, PENG Liang, ZENG Xian-zhu, ZHENG Da-gui
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16229
2017 Vol. 25 (2): 112-120 [
Abstract
] (
303
)
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(1 KB)
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(2358 KB) (
626
)
121
“One-Pot” Synthesis of
α,β
-Alkynones Promoted by Magnesium Powder
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.2.16264
2017 Vol. 25 (2): 121-126 [
Abstract
] (
282
)
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(1 KB)
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(663 KB) (
312
)
127
Synthesis of
p-
Methoxyacetophenone Catalyzed by Molecular Sieve PW-
β
/MCM-41 Modified with Phosphotungstic Acid
JIAO Lei, LIU Han, LI Hui-peng, ZHAO Hua
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16177
2017 Vol. 25 (2): 127-131 [
Abstract
] (
338
)
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(1 KB)
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(1485 KB) (
212
)
132
Hydrothermal Preparation of Chiolite-type Fluoride K
5
V
3
F
14
and Its Magnetic Property
HE Li-jie, ZHANG Dong, TAN Guang-lei, MU Tao, LIU Hai-yan, DU Peng
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16129
2017 Vol. 25 (2): 132-136 [
Abstract
] (
234
)
HTML
(1 KB)
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(1225 KB) (
251
)
137
Solid-phase Synthesis of Polypeptides BRC4 and Their Interaction with RAD51(231-260)
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16216
2017 Vol. 25 (2): 137-139 [
Abstract
] (
259
)
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(1 KB)
PDF
(470 KB) (
239
)
140
Preparation of A Novel Degradable Anti-inflammatory Sustain Release System By Combination of Hot Melt Extrusion and Electrospining Method
WANG Lian-song, YIN Li-li, LIU Dong, ZHENG Yu-qiang, HE Wei
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16175
2017 Vol. 25 (2): 140-143 [
Abstract
] (
280
)
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(1 KB)
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(811 KB) (
258
)
144
Synthesis of Methyl Laurate Catalyzed by Concerted Catalysis of TsOH Cooperate with I
2
WANG Lin-lin, DU Ying, WU Xiao-yun, LUO Shi-xia, YIN Xiao-gang
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16145
2017 Vol. 25 (2): 144-147 [
Abstract
] (
249
)
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(1 KB)
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(686 KB) (
204
)
148
Synthesis of An End-hydroxy PAMAM Molecular
SHI Jun, GUO Xiao-yi, WANG Ru-bin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16242
2017 Vol. 25 (2): 148-151 [
Abstract
] (
276
)
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(1 KB)
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(1004 KB) (
250
)
152
Analysis of Related Substances in The Production of Ursodeoxycholic Acid
XIE Qiang, WANG Kun, TAO Jia-lin
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16279
2017 Vol. 25 (2): 152-154 [
Abstract
] (
425
)
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(1 KB)
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(578 KB) (
295
)
155
Research on Selective Demethylation of Trimethoxybenzene Compounds
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16185
2017 Vol. 25 (2): 155-158 [
Abstract
] (
262
)
HTML
(1 KB)
PDF
(846 KB) (
274
)
159
Microwave Synthesis of 4,7,10-Tris(
tert
-butoxycarbonylmethyl)-1,4,7,10-tetraazacyclodo-decane-1-acetohydrazide
ZHOU Jin, YANG Hai-dong, SUN Hong-shun, LI Yu-long, JIANG Hong
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16234
2017 Vol. 25 (2): 159-162 [
Abstract
] (
257
)
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(1 KB)
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(1734 KB) (
312
)
163
Synthesis and Properties of Acrylamide/Methyl Acryloyl Oxygen Ethyl Dimethyl Ammonium Propyl Sulfonic Acid Copolymer
GUAN Hui-min, ZHAGN Wei-wei, YU Ting-yun
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16223
2017 Vol. 25 (2): 163-165 [
Abstract
] (
260
)
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(1 KB)
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(788 KB) (
280
)
166
Process Improvement on the Synthesis of Afatinib
LI Wen-qian, SONG Guo-qiang, WAN Yi-dong, GAO You-jun, FENG Xiao-qing
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16253
2017 Vol. 25 (2): 166-169 [
Abstract
] (
409
)
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(1 KB)
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(1343 KB) (
373
)
170
Process Improvement on Synthesis of Vitamin D
2
-A and CD Ring Fragment Alcohol
CHEN Guang-yao, BAO Xiao-zhen, DING Ying, ZHANG Heng-rui, FANG Zhi-jie
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16225
2017 Vol. 25 (2): 170-172 [
Abstract
] (
274
)
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(1 KB)
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(573 KB) (
244
)
173
Research Progress on Synthesis of Acridine Derivatives
WEI Qiang, GENG Xin-le
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16288
2017 Vol. 25 (2): 173-177 [
Abstract
] (
374
)
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(1 KB)
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(3739 KB) (
708
)
178
Research Progress on the Synthesis and Bioactivities of Indole-3-glyoxylamide Derivatives
HU Hong-yu, WANG Fei, ZHAO Sheng-xian, FANG Mei-juan
DOI: 10.15952/j.cnki.cjsc.1005-1511.2017.02.16207
2017 Vol. 25 (2): 178-184 [
Abstract
] (
362
)
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(1 KB)
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(2621 KB) (
263
)
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